静岡大学

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Researcher DataBase - Personal Information : NARUMI Tetsuo

Papers, etc.

【Papers, etc.】
[1]. Fine bubble technology for the green synthesis of fairy chemicals Org. Biomol. Chem. in press/ in press- (2024) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] A. K. Manna, M. Doi, K. Matsuo, H. Sakurai, C. Subrahamayam, K. Sato, T. Narumi, N. Mase [DOI] [2]. Late-Stage Derivatization of Oleanolic Acid-Based Anti-HIV-1 Compounds Chem. Pharm. Bull. 72/ 330-335 (2024) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Reon Takeuchi, Junko Fujimoto, Yoshinori Taguchi, Ryuji Ide, Ryuji Kyan, Kohei Sato, Nobuyuki Mase, Masaru Yokoyama, Shigeyoshi Harada, Tetsuo Narumi [DOI] [3]. Amide-to-Chloroalkene Substitution for Overcoming Intramolecular Acyl Transfer Challenges in Hexapeptidic Neuromedin U Receptor 2 Agonists Chemical Communications 60/ 3563-3566 (2024) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Tetsuo Narumi, Daichi Toyama, Junko Fujimoto, Ryuji Kyan, Kohei Sato, Kenji Mori, James T. Pearson, Nobuyuki Mase, Kentaro Takayama [DOI] [4]. Rapid identification of enamine-based organocatalysts for quaternary carbon-containing aldol reactions via fluorescence-based screening Asian J. Org. Chem. 12/ e202300236- (2023) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] H. Ito, Y. Yoshida, T. Masuda, A. Sasaki, K. Imoto, K. Sato, T. Narumi, N. Mase [DOI] [5]. Late-stage diversification strategy for the synthesis of peptide acids and amides using hydrazides Explor. Drug Sci. 1/ 322-335 (2023) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] S. Tanaka, M. Kanno, Y. Tashiro, T. Narumi, N. Mase, K. Sato [DOI] [6]. Enhancing Multiphase Reactions by Boosting Local Gas Concentration with Ultrafine Bubbles Bull. Chem. Soc. Jpn. 96/ 752-758 (2023) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] T. Kozuka, T. Iio, S. Suzuki, K. Kakiuchi, G. Tadano, K. Sato, T. Narumi, N. Mase [DOI] [7]. Design, synthesis, and bio-evaluation of novel triterpenoid derivatives as anti-HIV-1 compounds Bioorganic & Medicinal Chemistry Letters 69/1 128768-128773 (2022) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Reon Takeuchi, Kasumi Ogihara, Junko Fujimoto, Kohei Sato, Nobuyuki Mase, Kazuhisa Yoshimura, Shigeyoshi Harada, Tetsuo Narumi [DOI] [8]. Synthesis and structural characterization of β-turn mimics containing (Z)-chloroalkene dipeptide isosteres The Journal of Organic Chemistry 87/ 2167-2177 (2022) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Y. Kodama$$S. Takeo$$J. Fujimoto$$K. Sato$$N. Mase$$T. Narumi [DOI] [9]. β,γ-trans-selective γ-butyrolactone formation via homoenolate cross-annulation of enals and aldehydes catalyzed by sterically hindered N-heterocyclic carbene Tetrahedron 91/ 13219-13224 (2021) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] R. Kyan, Y. Kitagawa, R. Ide, K. Sato, N. Mase, T. Narumi [DOI] [10]. Stereoselective synthesis of highly functionalized (Z)-chloroalkene dipeptide isosteres containing an α,α-disubstituted amino acid Chemical Communications 57/ 6915-6918 (2021) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Y. Kodama$$S. Imai$$J. Fujimoto$$K. Sato$$N. Mase$$T. Narumi [DOI] [11]. Late-Stage Solubilization of Poorly Soluble Peptides Using Hydrazide Chemistry Organic Letters in press/ in press- (2021) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] Kohei Sato, Shoko Tanaka, Junzhen Wang, Kenya Ishikawa, Shugo Tsuda, Tetsuo Narumi, Taku Yoshiya, Nobuyuki Mase [DOI] [12]. Fine bubble–slug flow hydrogenation of multiple bonds and phenols Synlett / - (2020) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] Iio, T.$$Ngai, K.$$Kozuka, T.$$ Sammi, A. T.$$ Sato, K.$$, Narumi, T.$$Mase, N. [13]. Pendant Alkoxy Groups on N-Aryl Substitutions Drive the Efficiency of Imidazolylidene Catalysts for Homoenolate Annulation from Enal and Aldehyde Angewandte Chemie-International Edition 59/43 19031-19036 (2020) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Ryuji Kyan, Kohei Sato, Nobuyuki Mase, and Tetsuo Narumi [DOI] [14]. Stereoselective synthesis of Gly-Gly-type (E)- methylalkene and (Z)-chloroalkene dipeptide isosteres and their application to 14-mer RGG peptidomimetics RSC Advances 10/ 29373-29377 (2020) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Hikari Okita, Yuna Kato, Tatsuki Masuzawa, Kosuke Arai, Sayuri Takeo, Kohei Sato, Nobuyuki Mase, Takanori Oyoshi and Tetsuo Narumi [URL] [DOI] [15]. Chemoselective Umpolung of Enals for Asymmetric Homoenolate Cross-Annulation of Enals and Aldehydes Catalyzed by N-Heterocyclic Carbene Organic Letters 21/22 9119-9123 (2019) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Ryuji Ide, Ryuji Kyan, Kohei Sato, Nobuyuki Mase, Tetsuo Narum [DOI] [16]. Improvement of chemical stability of conjugated dienes by chlorine substitution Tetrahedron / - (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Tetsuo Narumi, Takuma Nishizawa, Tomoyuki Imai, Kohei Sato, Nobuyuki Mase [DOI] [17]. Novel Visible Light Photoactivatable Caged Neurotransmitter Based on a N-Methyl Quinolinium Chromophore YAKUGAKUZASSHI / - (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] 鳴海哲夫 [18]. Direct synthesis of N-terminal thiazolidine-containing peptide thioesters from peptide hydrazides Chem. Commun. / - (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] Kohei Sato, Shoko Tanaka, Kazuki Yamamoto, Yosuke Tashiro, Tetsuo Narumi, Nobuyuki Mase [DOI] [19]. 7-Hydroxy-N-Methylquinolinium Chromophore: A Photolabile Protecting Group for Blue Light Uncaging Organic Letters 20/14 4178-4182 (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Tetsuo Narumi, Koichi Miyata, Akitaka Nii, Kohei Sato, Nobuyuki Mase, Toshiaki Furuta [DOI] [20]. Organocatalytic Stereoselective Cyclic Polylactide Synthesis in Supercritical Carbon Dioxide under Plasticizing Conditions Polymers 10/ 713-722 (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] Nobuyuki Mase, Moniruzzaman, Shoji Yamamoto, Yoshitaka Nakaya, Kohei Sato, Tetsuo Narumi [DOI] [21]. The role of Chemisorption for Push-Pull Chromophores on SiO2 Surfaces in Non-Electrically Poling Host-Guest NLO Polymers J. Photochem. Photobiol., A: Chem. 340/1 35-45 (2017) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]杉田篤史 [共著者]間瀬暢之,佐藤浩平,田坂茂,川田善正,鳴海哲夫 [Notes] 合成担当 [22]. Tuning the Catalyst Reactivity of Imidazolylidene Catalysts through Substituent Effects on the N-Aryl Groups Org. Lett. 19/10 2750-2753 (2017) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] [責任著者]鳴海哲夫 [共著者]喜屋武龍二,佐藤浩平,間瀬暢之,渡辺修治 [23]. Fine-Bubble-Based Strategy for the Pd-Catalysed Hydrogenation of Nitro Groups: Measurement of Ultrafine Bubbles in Organic Solvents Synlett 28/16 2184-2188 (2017) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobuyuki Mase [共著者]Yuki Nishina,Shogo Isomura,Kohei Sato,Tetsuo Narumi,Naoharu Watanabe [24]. Microwave-Assisted Synthesis of Azacoumarin Fluorophores and the Fluorescence Characterization. The Journal of organic chemistry 82/5 2739-2744 (2017) [Refereed] non-refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Hikaru Takano,Tetsuo Narumi,Wataru Nomura [25]. Synthesis of a self-assembling gold nanoparticle-supported organocatalyst for enamine-based asymmetric aldol reactions Tetrahedron 72/16 1984-1990 (2016) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobuyuki Mase [共著者]Pe ter Lajos So ti,Hiroki Yamashita,Kohei Sato,Tetsuo Narumi,Mitsuo Toda [26]. Characteristic Fluctuations in Glycosidically Bound Volatiles during Tea Processing and Identification of Their Unstable Derivatives Journal of Agricultural and Food Chemistry 64/5 1151-1157 (2016) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Naoharu Watanabe,Huarong Tong [共著者]Jilai Cui,Toshiyuki Ohnishi,Nobuyuki Mase,Mitsuo Toda,Tetsuo Narumi [27]. A minimally cytotoxic CD4 mimic as an HIV entry inhibitor Bioorg Med Chem Lett 26/2 397-400 (2016) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Takaaki MIzuguchi,Shigeyoshi Harada,Tetsuo Narumi,Shuzo Matsushita,Kazuhisa Yoshimura,Hirokazu Tamamura [URL] [28]. Utilization of the Heavy Atom Effect for the Development of a Highly Photosensitive 8-Azacoumarin-type Photolabile Protecting Group Organic Letters 17/21 5372-5375 (2015) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] [責任著者]Tetsuo Narumi,Hirokazu Tamamura, [共著者]Hikaru Takano,Tetsuo Narumi,Wataru Nomura,Toshiaki Furuta,Hirokazu Tamamura [DOI] [29]. Remote Stereoinduction in the Organocuprate-Mediated Allylic Alkylation of Allylic gem-Dichlorides: Highly Diastereoselective Synthesis of (Z)-Chloroalkene Dipeptide Isosteres Organic Letters 17/10 2302-2305 (2015) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] author [Author] [責任著者]Tetsuo NARUMI,Hirokazu TAMAMURA [共著者]Takuya KOBAYAKAWA [DOI] [30]. Isostere-Based Design of 8-Azacoumarin-Type Photolabile Protecting Groups: A Hydrophilicity-Increasing Strategy for Coumarin-4-ylmethyls Org. Lett. 16/4 1184-1187 (2014) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Hikaru Takano,Nami Ohashi,Akinobu Suzuki,Toshiaki Furuta [DOI] [31]. Imidazolium Salt-Catalyzed Friedel-Crafts-Type Conjugate Addition of Indoles: Analysis of Indole/Imidazolium Complex by High Level ab Initio Calculations Asian Journal of Organic Chemistry 3/(num) (xxx) - (zzz) (2014) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Seiji Tsuzuki [32]. A CD4 Mimic as an HIV Entry Inhibitors: Pharmacokinetics Bioorg. Med. Chem. 21/24 7884-7889 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Chie Hashimoto,Tetsuo Narumi,Kazuhisa Yoshimura,Wataru Nomura,Shuzo Matsushita [URL] [33]. Generation of a Replication-competent Simian-human Immunodeficiency Virus, the Neutralisation Sensitivity of Which can be Enhanced in the Presence of a Small Molecule CD4 Mimic J. Gen. Virol. 94/(num) 2710-2716 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Tatsuhiko Igarashi [共著者]Hiroyuki Otsuki,Tomoyuki Miura,Tetsuo Narumi,Kazuhisa Yoshimura,Shuzo Matsushita [URL] [34]. Peptide-based Ligand Screening and Functional Analysis of Protein Kinase C Biopolymers: Peptide Science. 100/6 613-620 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Nami Ohashi,Wataru Nomura,Tetsuo Narumi,, [DOI] [35]. CD4 Mimics as HIV Entry Inhibitors: Lead Optimization Studies of the Aromatic Substituents Bioorg. Med. Chem. Lett. 21/9 2518-2526 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Hiroshi Arai,Kazuhisa Yoshimura,Shuzo Matsushita,Wataru Nomura [URL] [36]. Low Molecular Weight CXCR4 Ligands with Variable Spacers ChemMedChem. 8/1 118-124 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Haruo Aikawa,Tomohiro Tanaka,Tsutomu Murakami ,Naoki Yamamoto [DOI] [37]. Stereoselective Formation of Trisubstituted (Z)-Chloroalkenes Adjacent to a Tertiary Carbon Stereogenic Center by Organocuprate-Mediated Reduction/Alkylation Org. Lett. 14/17 4490-4493 (2012) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Takuya Kobayakawa,Haruo Aikawa,Shunsuke Seike, [DOI] [38]. Pharmacophore-Based Small Molecule CXCR4 Ligands Bioorg. Med. Chem. Lett. 22/15 4169-4172 (2012) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Tomohiro Tanaka,Wataru Nomura,Tsutomu Murakami,Haruo Aikawa [URL] [39]. Evaluation of a Synthetic C34 Trimer of HIV-1 gp41 as AIDS Vaccines Bioorg. Med. Chem. 20/10 3287-3291 (2012) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Chie Hashimoto,Wataru Nomura,Tetsuo Narumi,Haruo Aikawa,Naoki Yamamoto [URL] [40]. Conjugation of Cell-penetrating Peptides Leads to Identification of Anti-HIV Peptides from Matrix Proteins Bioorg. Med. Chem. 20/4 1468-1474 (2012) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Mao Komoriya,Wataru Nomura,Naoki Yamamoto ,Tsutomu Murakami [URL] [41]. Synthetic C34 Trimer of HIV-1 gp41 Shows Significant Increase of Inhibition Potency ChemMedChem. 7/2 205-208 (2012) [Refereed] non-refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Wataru Nomura,Chie Hashimoto,Tetsuo Narumi,Naoki Yamamoto, [DOI] [42]. α,α-Dichloroisoxazolidinones for the synthesis and chemoselective peptide ligation of α-peptide α-ketoacids Heterocycles 82/2 1515-1525 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Jeffrey W. Bode [共著者]Tetsuo Narumi [URL] [43]. Small Molecular CD4 Mimics as HIV Entry Inhibitors Bioorg. Med. Chem. 19/22 6735-6742 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Hiroshi Arai,Kazuhisa Yoshimura,Wataru Nomura,Shuzo Matsushita [URL] [44]. The Success and Failures of HIV Drug Discovery Expert Opin. Drug Discovery 6/10 1067-1090 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Chie Hashimoto,Tmohiro Tanaka,Tetsuo Narumi,Wataru Nomura [DOI] [45]. Fluorescence-Quenching Screening of Protein Kinase C Ligands with an Environmentally Sensitive Fluorophore Bioconjugate Chem. 22/5 923-930 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Wataru Nomura,Nami Ohashi,Tetsuo Narumi,Teikichi Ikura,Nobutoshi Ito [DOI] [46]. Azamacrocyclic-metal Complexes as CXCR4 Antagonists ChemMedChem 6/5 834-839 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] author [Author] [責任著者]Tetsuo Narumi,Hirokazu Tamamura [共著者]Tomohiro Tanaka,Wataru Nomura,Tsutomu Murakami,Naoki Yamamoto [DOI] [47]. Synthetic Caged DAG-lactones for Photochemically-controlled Activation of Protein Kinase C ChemBioChem 12/4 535-539 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Wataru Nomura,Tetsuo Narumi,Yuki Serizawa,Peter M. Blumberg,Toshiaki Furuta [DOI] [48]. Fluorescent-responsive Synthetic C1b Domains of Protein Kinase Cδ as Reporters of Specific High Affinity Ligand Binding Bioconjugate Chem. 22/1 82-87 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Nami Ohashi,Wataru Nomura,Tetsuo Narumi,Peter M. Blumberg, [DOI] [49]. Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres Org. Biomol. Chem. 8/(num) 616-621 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Shinya Oishi,Nobutaka Fujii [共著者]Tetsuo Narumi,Hiroaki Ohno,Takeshi Naito,Eiichi Kodama,Masao Matsuoka [URL] [50]. Bivalent Ligands of CXCR4 with Rigid Linkers for Elucidation of the Dimerization State in Cells J. Am. Chem. Soc. 132/(num) 15899-15901 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Wataru Nomura,Hirokazu Tamamura [共著者]Tomohiro Tanaka,Akemi Masuda,Tetsuo Narumi [DOI] [51]. CD4 mimics targeting the HIV entry mechanism and their hybrid molecules with a CXCR4 antagonist Bioorg. Med. Chem. Lett. 20/19 5853-5858 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Chihiro Ochiai,Kazuhisa Yoshimura,Wataru Nomura,Shuzo Matsushita [URL] [52]. Peptidic HIV integrase inhibitors derived from HIV gene products: structure-activity relationship studies Bioorg. Med. Chem. 18/18 6771-6775 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Shintaro Suzuki,Kasthuraiah Maddali,Hiroshi Tsutsumi,Tetsuo Narumi,Yves Pommier [URL] [53]. Development of crosslink-type tag-probe pairs for fluorescent imaging of proteins Biopolimers: Peptide Science 94/(num) 843-852 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Wataru Nomura,Tomoaki Mino,Tetsuo Narumi,Hiroshi Tsutsumi, [DOI] [54]. Peptide HIV-1 Integrase Inhibitors from HIV-1 Gene Products J. Med. Chem. 53/14 5356-5360 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Shintaro Suzuki,Kasthuraiah Maddali,Yves Pommier ,Tetsuo Narumi,Naoki Yamamoto [DOI] [55]. Remodeling of dynamic structures of HIV-1 envelope proteins leads to synthetic antigen molecules including neutralizing antibodies Bioconjugate Chem. 21/4 709-714 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Wataru Nomura,Hirokazu Tamamura [共著者]Toru Nakahara,Tetsuo Narumi,Tsutomu Murakami,Naoki Yamamoto, [DOI] [56]. CD4 mimics targeting the mechanism of HIV entry Bioorg. Med. Chem. Lett. 20/1 354-358 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Hirokazu Tamamura [共著者]Yuko Yamada,Kazuhisa Yoshimura,Tetsuo Narumi,Wataru Nomura,Shuzo Matsushita [DOI] [57]. Synthesis of protein kinase Cδ C1b domain by native chemical ligation methodology andcharacterization of its folding and ligand binding J. Pep. Sci. 15/(num) 626-646 (2009) [Refereed] non-refereed [Internationally co-authored papers] non-internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Wataru Nomura,Hirokazu Tamamura [共著者]Nami Ohashi,Tetsuo Narumi,Peter M. Blumberg, [URL] [58]. Structure-activity relationship study on artificial CXCR4 ligand possessing the cyclic pentapeptide scaffold: the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids Org. Biomol. Chem. 7/(num) 3805-3809 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Wataru Nomura,Hirokazu Tamamura [共著者]Tomohiro Tanaka,Tetsuo Narumi,Shinya Oishi,Stephen C. Peiper,Nobutaka Fujii [URL] [59]. Amino Acid-Based Synthesis of Trifluoromethylalkene Dipeptide Isosteres by Alcohol-Assisted Nucleophilic Trifluoromethylation and Organozinc-Copper-Mediated SN2’ Alkylation J. Org. Chem. 74/12 4626-4629 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobutaka Fujii [共著者]Kazuya Kobayashi,Tetsuo Narumi,Shinya Oishi,Hiroaki Ohno [DOI] [60]. eptide Bond Mimicry by (E)-Alkene and (Z)-Fluoroalkene Peptide Isosteres: Synthesis and Bioevaluation of α-Helical Anti-HIV Peptide Analogues Org. Biomol. Chem. 7/(num) 2872-2877 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Shinya Oishi,Nobutaka Fujii [共著者]Hirotaka Kamitani,Yasuyo Kodera,Tetsuo Narumi,Takeshi Naito,Masao Matsuoka [URL] [61]. Synthesis of Fluoroalkene Dipeptide Isosteres by an Intramolecular Redox Reaction Utilizing N-Heterocyclic Carbenes (NHCs) J. Org. Chem. 74/9 3272-3277 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Akira Otaka [共著者]Yoko Yamaki,Akira Shigenaga,Tetsuo Narumi,Nobutaka Fujii, [DOI] [62]. Synthesis and Application of (Z)-Alkene- and (E)-Fluoroalkene-Dipeptide Isosteres as cis-Amide Equivalents Adv. Exp. Med. Biol. 611/(num) 365-366 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobutaka Fujii [共著者]Kenji Tomita,Tetsuo Narumi,Ayumu Niida,Shinya Oishi,Hiroaki Ohno [DOI] [63]. Diastereoselective Synthesis of Highly Functionalized Fluoroalkene Dipeptide Isosteres and Its Application to Fmoc-Based Solid-Phase Synthesis of a Cyclic Pentapeptide Mimetic Tetrahedron 64/19 4332-4346 (2008) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobutaka Fujii [共著者]Tetsuo Narumi,kenji Tomita,Kazuya Kobayashi,Shinya Oishi,Hiroaki Ohno [DOI] [64]. Efficient Synthesis of Trifluoromethyl and Related Trisubstituted Alkene Dipeptide Isosteres by Palladium-Catalyzed Carbonylation of Amino Acid Derived Allylic Carbonates J. Org. Chem. 73/10 3942-3945 (2008) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobutaka Fujii [共著者]Eriko Inokuchi,Tetsuo Narumi,Ayumu Niida,Shinya Oishi,Hiroaki Ohno [DOI] [65]. Facile Synthesis of Fluoroalkenes by Palladium-Catalyzed Reductive Defluorination by Allylic gem-Difluorides Org. Lett. 9/(num) 3465-3468 (2007) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobutaka Fujii [共著者]Tetsuo Narumi,Kenji Tomita,Shinya Oishi,Hiroaki Ohno [DOI] [66]. Fmoc-Based Solid-Phase Synthesis of GPR54-Agonistic Pentapeptide Derivatives Containing Alkene- and Fluoroalkene-Dipeptide Isosteres Biopolymer 88/(num) 272-278 (2007) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobutaka Fujii [共著者]Kenji Tomita,Tetsuo Narumi,Akira Otaka,Shinya Oishi,Hiroaki Ohno [DOI] [67]. A Novel One-Pot Reaction Involving Organocopper-Mediated Reduction/ Transmetalation/Asymmetric Alkylation, Leading to the Diastereoselective Synthesis of Functionalized (Z)-Fluoroalkene Dipeptide Isosteres Chem. Commun. (vol)/(num) 4720-4722 (2006) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobutaka Fujii [共著者]Tetsuo Narumi,Shinya Oishi,Akira Otaka,Hiroaki Ohno [URL] [68]. Synthesis of (Z)-Alkene and (E)-Fluoroalkene Containing Diketopiperazine Mimetics Utilizing Organocopper-mediated Reduction-Alkylation and Diastereoselectivity Examination using DFT Calculations J. Org. Chem. 71/11 4118-4129 (2006) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper [Lead author or co-author] co-author [Author] [責任著者]Nobutaka Fujii [共著者]Ayumu Niida,Tetsuo Narumi,Hiroaki Ohno,Akira Otaka,Kazuo Kitaura [DOI]

[1]. Fine bubble technology for the green synthesis of fairy chemicals
Org. Biomol. Chem. in press/ in press- (2024) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] A. K. Manna, M. Doi, K. Matsuo, H. Sakurai, C. Subrahamayam, K. Sato, T. Narumi, N. Mase [DOI]
[2]. Late-Stage Derivatization of Oleanolic Acid-Based Anti-HIV-1 Compounds
Chem. Pharm. Bull. 72/ 330-335 (2024) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Reon Takeuchi, Junko Fujimoto, Yoshinori Taguchi, Ryuji Ide, Ryuji Kyan, Kohei Sato, Nobuyuki Mase, Masaru Yokoyama, Shigeyoshi Harada, Tetsuo Narumi [DOI]
[3]. Amide-to-Chloroalkene Substitution for Overcoming Intramolecular Acyl Transfer Challenges in Hexapeptidic Neuromedin U Receptor 2 Agonists
Chemical Communications 60/ 3563-3566 (2024) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Tetsuo Narumi, Daichi Toyama, Junko Fujimoto, Ryuji Kyan, Kohei Sato, Kenji Mori, James T. Pearson, Nobuyuki Mase, Kentaro Takayama [DOI]
[4]. Rapid identification of enamine-based organocatalysts for quaternary carbon-containing aldol reactions via fluorescence-based screening
Asian J. Org. Chem. 12/ e202300236- (2023) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] H. Ito, Y. Yoshida, T. Masuda, A. Sasaki, K. Imoto, K. Sato, T. Narumi, N. Mase [DOI]
[5]. Late-stage diversification strategy for the synthesis of peptide acids and amides using hydrazides
Explor. Drug Sci. 1/ 322-335 (2023) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] S. Tanaka, M. Kanno, Y. Tashiro, T. Narumi, N. Mase, K. Sato [DOI]
[6]. Enhancing Multiphase Reactions by Boosting Local Gas Concentration with Ultrafine Bubbles
Bull. Chem. Soc. Jpn. 96/ 752-758 (2023) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] T. Kozuka, T. Iio, S. Suzuki, K. Kakiuchi, G. Tadano, K. Sato, T. Narumi, N. Mase [DOI]
[7]. Design, synthesis, and bio-evaluation of novel triterpenoid derivatives as anti-HIV-1 compounds
Bioorganic & Medicinal Chemistry Letters 69/1 128768-128773 (2022) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Reon Takeuchi, Kasumi Ogihara, Junko Fujimoto, Kohei Sato, Nobuyuki Mase, Kazuhisa Yoshimura, Shigeyoshi Harada, Tetsuo Narumi [DOI]
[8]. Synthesis and structural characterization of β-turn mimics containing (Z)-chloroalkene dipeptide isosteres
The Journal of Organic Chemistry 87/ 2167-2177 (2022) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Y. Kodama$$S. Takeo$$J. Fujimoto$$K. Sato$$N. Mase$$T. Narumi [DOI]
[9]. β,γ-trans-selective γ-butyrolactone formation via homoenolate cross-annulation of enals and aldehydes catalyzed by sterically hindered N-heterocyclic carbene
Tetrahedron 91/ 13219-13224 (2021) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] R. Kyan, Y. Kitagawa, R. Ide, K. Sato, N. Mase, T. Narumi [DOI]
[10]. Stereoselective synthesis of highly functionalized (Z)-chloroalkene dipeptide isosteres containing an α,α-disubstituted amino acid
Chemical Communications 57/ 6915-6918 (2021) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Y. Kodama$$S. Imai$$J. Fujimoto$$K. Sato$$N. Mase$$T. Narumi [DOI]
[11]. Late-Stage Solubilization of Poorly Soluble Peptides Using Hydrazide Chemistry
Organic Letters in press/ in press- (2021) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] Kohei Sato, Shoko Tanaka, Junzhen Wang, Kenya Ishikawa, Shugo Tsuda, Tetsuo Narumi, Taku Yoshiya, Nobuyuki Mase [DOI]
[12]. Fine bubble–slug flow hydrogenation of multiple bonds and phenols
Synlett / - (2020) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] Iio, T.$$Ngai, K.$$Kozuka, T.$$ Sammi, A. T.$$ Sato, K.$$, Narumi, T.$$Mase, N.
[13]. Pendant Alkoxy Groups on N-Aryl Substitutions Drive the Efficiency of Imidazolylidene Catalysts for Homoenolate Annulation from Enal and Aldehyde
Angewandte Chemie-International Edition 59/43 19031-19036 (2020) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Ryuji Kyan, Kohei Sato, Nobuyuki Mase, and Tetsuo Narumi [DOI]
[14]. Stereoselective synthesis of Gly-Gly-type (E)- methylalkene and (Z)-chloroalkene dipeptide isosteres and their application to 14-mer RGG peptidomimetics
RSC Advances 10/ 29373-29377 (2020) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Hikari Okita, Yuna Kato, Tatsuki Masuzawa, Kosuke Arai, Sayuri Takeo, Kohei Sato, Nobuyuki Mase, Takanori Oyoshi and Tetsuo Narumi [URL] [DOI]
[15]. Chemoselective Umpolung of Enals for Asymmetric Homoenolate Cross-Annulation of Enals and Aldehydes Catalyzed by N-Heterocyclic Carbene
Organic Letters 21/22 9119-9123 (2019) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Ryuji Ide, Ryuji Kyan, Kohei Sato, Nobuyuki Mase, Tetsuo Narum [DOI]
[16]. Improvement of chemical stability of conjugated dienes by chlorine substitution
Tetrahedron / - (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Tetsuo Narumi, Takuma Nishizawa, Tomoyuki Imai, Kohei Sato, Nobuyuki Mase [DOI]
[17]. Novel Visible Light Photoactivatable Caged Neurotransmitter Based on a N-Methyl Quinolinium Chromophore
YAKUGAKUZASSHI / - (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] 鳴海哲夫
[18]. Direct synthesis of N-terminal thiazolidine-containing peptide thioesters from peptide hydrazides
Chem. Commun. / - (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] Kohei Sato, Shoko Tanaka, Kazuki Yamamoto, Yosuke Tashiro, Tetsuo Narumi, Nobuyuki Mase [DOI]
[19]. 7-Hydroxy-N-Methylquinolinium Chromophore: A Photolabile Protecting Group for Blue Light Uncaging
Organic Letters 20/14 4178-4182 (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Tetsuo Narumi, Koichi Miyata, Akitaka Nii, Kohei Sato, Nobuyuki Mase, Toshiaki Furuta [DOI]
[20]. Organocatalytic Stereoselective Cyclic Polylactide Synthesis in Supercritical Carbon Dioxide under Plasticizing Conditions
Polymers 10/ 713-722 (2018) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] Nobuyuki Mase, Moniruzzaman, Shoji Yamamoto, Yoshitaka Nakaya, Kohei Sato, Tetsuo Narumi [DOI]
[21]. The role of Chemisorption for Push-Pull Chromophores on SiO2 Surfaces in Non-Electrically Poling Host-Guest NLO Polymers
J. Photochem. Photobiol., A: Chem. 340/1 35-45 (2017) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]杉田篤史 [共著者]間瀬暢之,佐藤浩平,田坂茂,川田善正,鳴海哲夫 [Notes] 合成担当
[22]. Tuning the Catalyst Reactivity of Imidazolylidene Catalysts through Substituent Effects on the N-Aryl Groups
Org. Lett. 19/10 2750-2753 (2017) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] [責任著者]鳴海哲夫 [共著者]喜屋武龍二,佐藤浩平,間瀬暢之,渡辺修治
[23]. Fine-Bubble-Based Strategy for the Pd-Catalysed Hydrogenation of Nitro Groups: Measurement of Ultrafine Bubbles in Organic Solvents
Synlett 28/16 2184-2188 (2017) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobuyuki Mase [共著者]Yuki Nishina,Shogo Isomura,Kohei Sato,Tetsuo Narumi,Naoharu Watanabe
[24]. Microwave-Assisted Synthesis of Azacoumarin Fluorophores and the Fluorescence Characterization.
The Journal of organic chemistry 82/5 2739-2744 (2017) [Refereed] non-refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Hikaru Takano,Tetsuo Narumi,Wataru Nomura
[25]. Synthesis of a self-assembling gold nanoparticle-supported organocatalyst for enamine-based asymmetric aldol reactions
Tetrahedron 72/16 1984-1990 (2016) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobuyuki Mase [共著者]Pe ter Lajos So ti,Hiroki Yamashita,Kohei Sato,Tetsuo Narumi,Mitsuo Toda
[26]. Characteristic Fluctuations in Glycosidically Bound Volatiles during Tea Processing and Identification of Their Unstable Derivatives
Journal of Agricultural and Food Chemistry 64/5 1151-1157 (2016) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Naoharu Watanabe,Huarong Tong [共著者]Jilai Cui,Toshiyuki Ohnishi,Nobuyuki Mase,Mitsuo Toda,Tetsuo Narumi
[27]. A minimally cytotoxic CD4 mimic as an HIV entry inhibitor
Bioorg Med Chem Lett 26/2 397-400 (2016) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Takaaki MIzuguchi,Shigeyoshi Harada,Tetsuo Narumi,Shuzo Matsushita,Kazuhisa Yoshimura,Hirokazu Tamamura [URL]
[28]. Utilization of the Heavy Atom Effect for the Development of a Highly Photosensitive 8-Azacoumarin-type Photolabile Protecting Group
Organic Letters 17/21 5372-5375 (2015) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] [責任著者]Tetsuo Narumi,Hirokazu Tamamura, [共著者]Hikaru Takano,Tetsuo Narumi,Wataru Nomura,Toshiaki Furuta,Hirokazu Tamamura [DOI]
[29]. Remote Stereoinduction in the Organocuprate-Mediated Allylic Alkylation of Allylic gem-Dichlorides: Highly Diastereoselective Synthesis of (Z)-Chloroalkene Dipeptide Isosteres
Organic Letters 17/10 2302-2305 (2015) [Refereed] refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] author
[Author] [責任著者]Tetsuo NARUMI,Hirokazu TAMAMURA [共著者]Takuya KOBAYAKAWA [DOI]
[30]. Isostere-Based Design of 8-Azacoumarin-Type Photolabile Protecting Groups: A Hydrophilicity-Increasing Strategy for Coumarin-4-ylmethyls
Org. Lett. 16/4 1184-1187 (2014) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Hikaru Takano,Nami Ohashi,Akinobu Suzuki,Toshiaki Furuta [DOI]
[31]. Imidazolium Salt-Catalyzed Friedel-Crafts-Type Conjugate Addition of Indoles: Analysis of Indole/Imidazolium Complex by High Level ab Initio Calculations
Asian Journal of Organic Chemistry 3/(num) (xxx) - (zzz) (2014) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Seiji Tsuzuki
[32]. A CD4 Mimic as an HIV Entry Inhibitors: Pharmacokinetics
Bioorg. Med. Chem. 21/24 7884-7889 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Chie Hashimoto,Tetsuo Narumi,Kazuhisa Yoshimura,Wataru Nomura,Shuzo Matsushita [URL]
[33]. Generation of a Replication-competent Simian-human Immunodeficiency Virus, the Neutralisation Sensitivity of Which can be Enhanced in the Presence of a Small Molecule CD4 Mimic
J. Gen. Virol. 94/(num) 2710-2716 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Tatsuhiko Igarashi [共著者]Hiroyuki Otsuki,Tomoyuki Miura,Tetsuo Narumi,Kazuhisa Yoshimura,Shuzo Matsushita [URL]
[34]. Peptide-based Ligand Screening and Functional Analysis of Protein Kinase C
Biopolymers: Peptide Science. 100/6 613-620 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Nami Ohashi,Wataru Nomura,Tetsuo Narumi,, [DOI]
[35]. CD4 Mimics as HIV Entry Inhibitors: Lead Optimization Studies of the Aromatic Substituents
Bioorg. Med. Chem. Lett. 21/9 2518-2526 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Hiroshi Arai,Kazuhisa Yoshimura,Shuzo Matsushita,Wataru Nomura [URL]
[36]. Low Molecular Weight CXCR4 Ligands with Variable Spacers
ChemMedChem. 8/1 118-124 (2013) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Haruo Aikawa,Tomohiro Tanaka,Tsutomu Murakami ,Naoki Yamamoto [DOI]
[37]. Stereoselective Formation of Trisubstituted (Z)-Chloroalkenes Adjacent to a Tertiary Carbon Stereogenic Center by Organocuprate-Mediated Reduction/Alkylation
Org. Lett. 14/17 4490-4493 (2012) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Takuya Kobayakawa,Haruo Aikawa,Shunsuke Seike, [DOI]
[38]. Pharmacophore-Based Small Molecule CXCR4 Ligands
Bioorg. Med. Chem. Lett. 22/15 4169-4172 (2012) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Tomohiro Tanaka,Wataru Nomura,Tsutomu Murakami,Haruo Aikawa [URL]
[39]. Evaluation of a Synthetic C34 Trimer of HIV-1 gp41 as AIDS Vaccines
Bioorg. Med. Chem. 20/10 3287-3291 (2012) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Chie Hashimoto,Wataru Nomura,Tetsuo Narumi,Haruo Aikawa,Naoki Yamamoto [URL]
[40]. Conjugation of Cell-penetrating Peptides Leads to Identification of Anti-HIV Peptides from Matrix Proteins
Bioorg. Med. Chem. 20/4 1468-1474 (2012) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Mao Komoriya,Wataru Nomura,Naoki Yamamoto ,Tsutomu Murakami [URL]
[41]. Synthetic C34 Trimer of HIV-1 gp41 Shows Significant Increase of Inhibition Potency
ChemMedChem. 7/2 205-208 (2012) [Refereed] non-refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Wataru Nomura,Chie Hashimoto,Tetsuo Narumi,Naoki Yamamoto, [DOI]
[42]. α,α-Dichloroisoxazolidinones for the synthesis and chemoselective peptide ligation of α-peptide α-ketoacids
Heterocycles 82/2 1515-1525 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Jeffrey W. Bode [共著者]Tetsuo Narumi [URL]
[43]. Small Molecular CD4 Mimics as HIV Entry Inhibitors
Bioorg. Med. Chem. 19/22 6735-6742 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Hiroshi Arai,Kazuhisa Yoshimura,Wataru Nomura,Shuzo Matsushita [URL]
[44]. The Success and Failures of HIV Drug Discovery
Expert Opin. Drug Discovery 6/10 1067-1090 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Chie Hashimoto,Tmohiro Tanaka,Tetsuo Narumi,Wataru Nomura [DOI]
[45]. Fluorescence-Quenching Screening of Protein Kinase C Ligands with an Environmentally Sensitive Fluorophore
Bioconjugate Chem. 22/5 923-930 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Wataru Nomura,Nami Ohashi,Tetsuo Narumi,Teikichi Ikura,Nobutoshi Ito [DOI]
[46]. Azamacrocyclic-metal Complexes as CXCR4 Antagonists
ChemMedChem 6/5 834-839 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] author
[Author] [責任著者]Tetsuo Narumi,Hirokazu Tamamura [共著者]Tomohiro Tanaka,Wataru Nomura,Tsutomu Murakami,Naoki Yamamoto [DOI]
[47]. Synthetic Caged DAG-lactones for Photochemically-controlled Activation of Protein Kinase C
ChemBioChem 12/4 535-539 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Wataru Nomura,Tetsuo Narumi,Yuki Serizawa,Peter M. Blumberg,Toshiaki Furuta [DOI]
[48]. Fluorescent-responsive Synthetic C1b Domains of Protein Kinase Cδ as Reporters of Specific High Affinity Ligand Binding
Bioconjugate Chem. 22/1 82-87 (2011) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Nami Ohashi,Wataru Nomura,Tetsuo Narumi,Peter M. Blumberg, [DOI]
[49]. Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres
Org. Biomol. Chem. 8/(num) 616-621 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Shinya Oishi,Nobutaka Fujii [共著者]Tetsuo Narumi,Hiroaki Ohno,Takeshi Naito,Eiichi Kodama,Masao Matsuoka [URL]
[50]. Bivalent Ligands of CXCR4 with Rigid Linkers for Elucidation of the Dimerization State in Cells
J. Am. Chem. Soc. 132/(num) 15899-15901 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Wataru Nomura,Hirokazu Tamamura [共著者]Tomohiro Tanaka,Akemi Masuda,Tetsuo Narumi [DOI]
[51]. CD4 mimics targeting the HIV entry mechanism and their hybrid molecules with a CXCR4 antagonist
Bioorg. Med. Chem. Lett. 20/19 5853-5858 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Tetsuo Narumi,Chihiro Ochiai,Kazuhisa Yoshimura,Wataru Nomura,Shuzo Matsushita [URL]
[52]. Peptidic HIV integrase inhibitors derived from HIV gene products: structure-activity relationship studies
Bioorg. Med. Chem. 18/18 6771-6775 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Shintaro Suzuki,Kasthuraiah Maddali,Hiroshi Tsutsumi,Tetsuo Narumi,Yves Pommier [URL]
[53]. Development of crosslink-type tag-probe pairs for fluorescent imaging of proteins
Biopolimers: Peptide Science 94/(num) 843-852 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Wataru Nomura,Tomoaki Mino,Tetsuo Narumi,Hiroshi Tsutsumi, [DOI]
[54]. Peptide HIV-1 Integrase Inhibitors from HIV-1 Gene Products
J. Med. Chem. 53/14 5356-5360 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Shintaro Suzuki,Kasthuraiah Maddali,Yves Pommier ,Tetsuo Narumi,Naoki Yamamoto [DOI]
[55]. Remodeling of dynamic structures of HIV-1 envelope proteins leads to synthetic antigen molecules including neutralizing antibodies
Bioconjugate Chem. 21/4 709-714 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Wataru Nomura,Hirokazu Tamamura [共著者]Toru Nakahara,Tetsuo Narumi,Tsutomu Murakami,Naoki Yamamoto, [DOI]
[56]. CD4 mimics targeting the mechanism of HIV entry
Bioorg. Med. Chem. Lett. 20/1 354-358 (2010) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Hirokazu Tamamura [共著者]Yuko Yamada,Kazuhisa Yoshimura,Tetsuo Narumi,Wataru Nomura,Shuzo Matsushita [DOI]
[57]. Synthesis of protein kinase Cδ C1b domain by native chemical ligation methodology andcharacterization of its folding and ligand binding
J. Pep. Sci. 15/(num) 626-646 (2009) [Refereed] non-refereed [Internationally co-authored papers] non-internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Wataru Nomura,Hirokazu Tamamura [共著者]Nami Ohashi,Tetsuo Narumi,Peter M. Blumberg, [URL]
[58]. Structure-activity relationship study on artificial CXCR4 ligand possessing the cyclic pentapeptide scaffold: the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids
Org. Biomol. Chem. 7/(num) 3805-3809 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Wataru Nomura,Hirokazu Tamamura [共著者]Tomohiro Tanaka,Tetsuo Narumi,Shinya Oishi,Stephen C. Peiper,Nobutaka Fujii [URL]
[59]. Amino Acid-Based Synthesis of Trifluoromethylalkene Dipeptide Isosteres by Alcohol-Assisted Nucleophilic Trifluoromethylation and Organozinc-Copper-Mediated SN2’ Alkylation
J. Org. Chem. 74/12 4626-4629 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobutaka Fujii [共著者]Kazuya Kobayashi,Tetsuo Narumi,Shinya Oishi,Hiroaki Ohno [DOI]
[60]. eptide Bond Mimicry by (E)-Alkene and (Z)-Fluoroalkene Peptide Isosteres: Synthesis and Bioevaluation of α-Helical Anti-HIV Peptide Analogues
Org. Biomol. Chem. 7/(num) 2872-2877 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Shinya Oishi,Nobutaka Fujii [共著者]Hirotaka Kamitani,Yasuyo Kodera,Tetsuo Narumi,Takeshi Naito,Masao Matsuoka [URL]
[61]. Synthesis of Fluoroalkene Dipeptide Isosteres by an Intramolecular Redox Reaction Utilizing N-Heterocyclic Carbenes (NHCs)
J. Org. Chem. 74/9 3272-3277 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Akira Otaka [共著者]Yoko Yamaki,Akira Shigenaga,Tetsuo Narumi,Nobutaka Fujii, [DOI]
[62]. Synthesis and Application of (Z)-Alkene- and (E)-Fluoroalkene-Dipeptide Isosteres as cis-Amide Equivalents
Adv. Exp. Med. Biol. 611/(num) 365-366 (2009) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobutaka Fujii [共著者]Kenji Tomita,Tetsuo Narumi,Ayumu Niida,Shinya Oishi,Hiroaki Ohno [DOI]
[63]. Diastereoselective Synthesis of Highly Functionalized Fluoroalkene Dipeptide Isosteres and Its Application to Fmoc-Based Solid-Phase Synthesis of a Cyclic Pentapeptide Mimetic
Tetrahedron 64/19 4332-4346 (2008) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobutaka Fujii [共著者]Tetsuo Narumi,kenji Tomita,Kazuya Kobayashi,Shinya Oishi,Hiroaki Ohno [DOI]
[64]. Efficient Synthesis of Trifluoromethyl and Related Trisubstituted Alkene Dipeptide Isosteres by Palladium-Catalyzed Carbonylation of Amino Acid Derived Allylic Carbonates
J. Org. Chem. 73/10 3942-3945 (2008) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobutaka Fujii [共著者]Eriko Inokuchi,Tetsuo Narumi,Ayumu Niida,Shinya Oishi,Hiroaki Ohno [DOI]
[65]. Facile Synthesis of Fluoroalkenes by Palladium-Catalyzed Reductive Defluorination by Allylic gem-Difluorides
Org. Lett. 9/(num) 3465-3468 (2007) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobutaka Fujii [共著者]Tetsuo Narumi,Kenji Tomita,Shinya Oishi,Hiroaki Ohno [DOI]
[66]. Fmoc-Based Solid-Phase Synthesis of GPR54-Agonistic Pentapeptide Derivatives Containing Alkene- and Fluoroalkene-Dipeptide Isosteres
Biopolymer 88/(num) 272-278 (2007) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobutaka Fujii [共著者]Kenji Tomita,Tetsuo Narumi,Akira Otaka,Shinya Oishi,Hiroaki Ohno [DOI]
[67]. A Novel One-Pot Reaction Involving Organocopper-Mediated Reduction/ Transmetalation/Asymmetric Alkylation, Leading to the Diastereoselective Synthesis of Functionalized (Z)-Fluoroalkene Dipeptide Isosteres
Chem. Commun. (vol)/(num) 4720-4722 (2006) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobutaka Fujii [共著者]Tetsuo Narumi,Shinya Oishi,Akira Otaka,Hiroaki Ohno [URL]
[68]. Synthesis of (Z)-Alkene and (E)-Fluoroalkene Containing Diketopiperazine Mimetics Utilizing Organocopper-mediated Reduction-Alkylation and Diastereoselectivity Examination using DFT Calculations
J. Org. Chem. 71/11 4118-4129 (2006) [Refereed] refereed [Internationally co-authored papers] internationally co-authored paper
[Lead author or co-author] co-author
[Author] [責任著者]Nobutaka Fujii [共著者]Ayumu Niida,Tetsuo Narumi,Hiroaki Ohno,Akira Otaka,Kazuo Kitaura [DOI]